| Name | CAS No. |
| Adagrasib / MRTX-819 | |
| Tert-Butyl 2,4-dichloro-5,6-dihydroxyprolido[3,4-d]pyrimidine-7(8H)-carboxylate | 916420-27-4 |
| (S)-2-(piperazin-2-yl)acetonitrile dihydrochloride | 2158301-19-8 |
| Atrasentan | |
| N-2 | 178739-03-2 |
| Ethyl 3-(4-methoxyphenyl)-3-oxopropionate | 2881-83-6 |
| Ethyl 3-(4-methoxyphenyl)-3-oxopropionate | 2881-83-6 |
| 2-Bromo-N,N-dibutylacetamide | 40124-27-4 |
| Baxdrostat | |
| 6-Bromo-1-methyl-1,2,3,4-tetrahydroquinolin-2-one | 1092523-03-9 |
| 1-Methyl-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-3,4-dihydroquinolin-2(1H)-one | 1427587-32-3 |
| (R)-4-Bromo-5,6,7,8-tetrahydroisoquinolin-8-amine | 1428652-00-9 |
| Brenoscatib VJ07986 | |
| (S)-4-(tert-butoxycarbonyl)-1,4-oxazepane-2-carboxylic acid | 1273567-44-4 |
| (S)-tert-butyl (1-amino-3-(4-iodophenyl)-1-oxopropan-2-yl)carbamate | 868694-44-4 |
| 3-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzol[dioxazol-2(3H)-one | 1220696-32-1 |
| Daraxonrasib / RMC-6236 | |
| (4-Bromophenyl)hydrazine hydrochloride | 41931-18-4 |
| 1-(3-Bromopyridin-2-yl)ethanone | 111043-09-5 |
| Methyl 5-chloro-2,2-dimethyl-5-oxopentanoatet | 98559-84-3 |
| Daridorexant | |
| (S)-2-Methylpyrrolidine-2-carboxylic acid hydrochloride | 1508261-86-6 |
| (2S)-Methyl 2-methylpyrrolidine-2-carboxylate hydrochloride | 220060-08-2 |
| 4-Chloro-3-methylbenzene-1,2-diamine hydrochloride-11 | 1087743-89-2 |
| 5-Methoxy-2-(2H-1,2,3-triazol-2-yl)benzoic acid-21 | 1293284-55-5 |
| Elinazentant | |
| 6-Chloro-4-(4-fluoro-2-methylphenyl)pyridin-3-amine hydrochloride | 2642577-31-7 |
| 2-[3,5-Bis(trifluoromethyl)phenyl]-2-methylpropanoic acid | 289686-70-0 |
| (7S,9aS)-7-((Benzyloxy)methyl)octahydropyrazino[2,1-c][1,4]oxazine dioxalate | 1268364-46-0 |
| Gepotidacin | |
| (S)-(3,8-Dioxo-1,2-dihydro-3H,8H-2a,5,8a-triazaacenaphthenyl-2-yl)methyl methanesulfonate | 2169933-17-7 |
| 3,4-Dihydro-2H-pyrano[2,3-c]pyridine-6-carbaldehyde | 527681-61-4 |
| Lazertinib | |
| 3-Phenyl-1H-pyrazole-4-carbaldehyde | 26033-20-5 |
| N-2 | 1903010-39-8 |
| Enlicitide Decanoate MK0616 | |
| 5-Fluoroidole | 399-52-0 |
| 5-Fluoro-L-tryptophan | 16626-02-1 |
| Boc-Tyr(Me)-OH | 53267-93-9 |
| Cbz-trans-3-Hydroxy-L-proline | 62182-54-1 |
| FMOC-D-DAP(Z)-OH | 387824-80-8 |
| Icotrokinra/JNJ-2113 | |
| 7-Methylindole | 933-67-5 |
| 2-Naphthaldehyde | 66-99-9 |
| L-Penicillamine | 1113-41-3 |
| Nerandomilast / BI-1015550 | |
| 2,4-dichloro-6,7-dihydrothieno[3,2-d]pyrimidine | 74901-69-2 |
| (1-Aminocyclobutyl)methanol hydrochloride | 1392213-15-8 |
| N-2 | 1423719-36-1 |
| 5-chloro-2-(piperidin-4-yl)pyrimidine hydrochloride | 1402666-88-9 |
| Renibrutinib | |
| 5-Fluoro-2-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline | 1418128-33-2 |
| tert-Butyl (2-((4-amino-6-chloropyrimidin-5-yl)oxy)ethyl)(methyl)carbamate | 1787294-51-2 |
| N-2 | 1787294-47-6 |
| Sparsentan | |
| 4,5-Dimethylisoxazol-3-amine | 13999-39-8 |
| N-2 | 415697-56-2 |
| Zastaprazan JP-1366 | |
| 5,6-Diamino-nicotinic acid methyl ester | 104685-76-9 |
| Seladepar | |
| Ethyl 2-(2-methylphenoxy)acetate | 93917-68-1 |
| Ethyl (4-mercapto-2-methylphenoxy)acetate | 343322-82-7 |
| (S)-2-((4-(Trifluoromethyl)phenoxy)methyl)oxirane | 256372-58-4 |
| Suzetrigine VX-518 | |
| Methyl 4-aminopyridine-2-carboxylate | 71469-93-7 |
| 2-(3,4-Difluoro-2-methoxyphenyl)acetic acid | 1558274-26-2 |
| N-4 | 2649470-89-1 |
| Xanomeline | |
| 3-Chloro-4-(pyridin-3-yl)-1,2,5-thiadiazole | 131986-28-2 |
| 3-(Hexyloxy)-4-(pyridin-3-yl)-1,2,5-thiadiazole | 131987-69-4 |